平安! 发表于 2011-11-9 19:57 ( K7 T. l$ Q8 b3 D# ?: `. v* F& d4 K
Pazopanib (100 mg/kg/day free base equivalent) 8 @, E$ X9 Q2 z$ n& b- Z2 F
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。9 v3 U# U; V. k& `. [
搜索了一下,原料一大堆。
+ T4 P5 ]6 g' }: t7 T
7 ?) f# a& J$ n- U" `$ y对不起!100mg/kg是用于移植瘤的,我弄错了。' i9 T9 h% t; h# l9 t! `9 m
. N/ E' \+ V/ d! G6 R# t; h以下是正版说明书的推荐用量。$ u+ o0 k- o2 Z; x+ d p+ r
1 s2 f( @; ~3 P. [& B+ b
--------------------- DOSAGE AND ADMINISTRATION ----------------
2 G% v; H4 c( a7 C* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) & ~2 W1 u8 ^/ G2 K" C
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
1 f& M" V k) g4 s+ T; g5 [1 p---------------------DOSAGE FORMS AND STRENGTHS --------------
. E9 J% Q5 X- Q( J/ K2 I200 mg tablets. (3)
. j% \, p2 j' |! _, i-------------------------------CONTRAINDICATIONS------------------------ |